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receptor artery migraine effect antagonist response study headache pharmacol agonist pacap vasodilatation blood telcagepant treatment segment sumatriptan antimigraine peptide concentration tegaserod vessel contraction trigeminal calcitonin gene-related peptide meningeal patient antimigraine drugs cgrp receptor antagonists mechanism model stimulation cephalalgia chapter triptan edvinsson cranial dural calcitonin panel 5- ht glutamate activation release figure heart gene-related pharmacology system right expression artery segments presence concentration response curves brain value meningeal arteries curve pac 1 receptor action experiment level relaxation increase nerve goadsby br j pharmacol blood vessels saxena pathophysiology vasoconstriction diameter nitric absence pacap 38 plasma ischemia glutamate receptor antagonists capsaicin contractile
9 Most Recent Publications
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Potential mechanisms of prospective antimigraine drugs: A focus on vascular (side) effects
(Article)
Chan, K.Y. Vermeersch, S. Hoon, J.N. de Villalón, C.M. MaassenVanDenBrink, A. |
2011-03-01
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Pharmacological characterization of VIP and PACAP receptors in the human meningeal and coronary artery
(Article)
Chan, K.Y. Baun, M. Gupta, S. Vries, R. de Bogaerdt, A. van den Dirven, C.M.F. Danser, A.H.J. Jansen-Olesen, I. Olesen, J. Villalón, C.M. MaassenVanDenBrink, A. |
2011-02-01
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Neurovascular Pharmacology of Prospective Antimigraine Drugs
(Doctoral Thesis)
Chan, K.Y. |
2011-01-26
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Effect of the calcitonin gene-related peptide (CGRP) receptor antagonist telcagepant in human cranial arteries
(Article)
Edvinsson, L. Chan, K.Y. Eftekhari, S. Nilsson, E. Vries, R. de Säveland, H. Dirven, C.M.F. Danser, A.H.J. |
2010-10-01
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Characterization of the calcitonin gene-related peptide receptor antagonist telcagepant (MK-0974) in human isolated coronary arteries
(Article)
Chan, K.Y. Edvinsson, L. Danser, A.H.J. MaassenVanDenBrink, A. Eftekhari, S. Kimblad, P.O. Kane, S.A. Lynch, J. Hargreaves, R.J. Vries, R. de Garrelds, I.M. Bogaerdt, A. van den |
2010-09-01
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Effects of ionotropic glutamate receptor antagonists on rat dural artery diameter in an intravital microscopy model
(Article)
Chan, K.Y. Gupta, S. Vries, R. de Danser, A.H.J. Villalón, C.M. Muñoz-Islas, E. Maassen van den Brink, A. |
2010-07-01
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Functional characterization of contractions to tegaserod in human isolated proximal and distal coronary arteries
(Article)
Chan, K.Y. Vries, R. de Leijten, F.P.J. Pfannkuche, H.J. Bogaerdt, A. van den Danser, A.H.J. MaassenVanDenBrink, A. |
2009-10-01
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Current and prospective pharmacological targets in relation to antimigraine action
(Article)
Mehrotra, S. Gupta, S. Chan, K.Y. Villalón, C.M. Centurion, D. Saxena, P.R. Maassen van den Brink, A. |
2008-10-01
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Neurovascular pharmacology of migraine
(Article)
MaassenVanDenBrink, A. Chan, K.Y. |
2008-05-13
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