In this thesis, several novel radiolabeled gastrin analogs were developed preclinically in vitro as well as in vivo in animal models.
In addition, the effect of in situ enzyme inhibition on metabolic stability and tumor uptake of the same gastrin radioligands was investigated.

M. de Jong (Marion) , T. Maina (Theodosia) , B.A. Nock (Berthold)
Erasmus University Rotterdam
hdl.handle.net/1765/93109
Erasmus MC: University Medical Center Rotterdam

Kaloudi, K. (2016, July 5). Radiolabeled gastrins in CCK2R-positive tumor targeting: Toward improved diagnostic efficacy via in situ enzyme-inhibition approaches. Retrieved from http://hdl.handle.net/1765/93109